Weight management, appetite regulation, blood sugar control, insulin level regulation, fat loss while preserving lean mass
Semaglutide es un agonista del receptor GLP-1 que imita la hormona incretina natural del cuerpo para ayudar a regular el apetito, el azúcar en sangre y los niveles de insulina. Se usa ampliamente para el control del peso y la salud metabólica debido a su capacidad para reducir el hambre, retardar el vaciado gástrico y favorecer la pérdida de grasa mientras se preserva la masa magra.
Mechanism of Action - Weight Management / Metabolic Pathway
Dosis inicial:0,25 mg una vez a la semana
Valoración:Aumentar gradualmente en 0,25-0,5 mg cada 2-4 semanas
Rango de mantenimiento típico:1 mg-2,5 mg por semana
| Period | Dose | Phase | Clinical Notes |
|---|---|---|---|
| Starting Dose | 0.25mg once weekly | initiation | Initial dose for treatment initiation |
| Titration | Increase by 0.25-0.5mg every 2-4 weeks | escalation | Gradual increase as tolerated |
| Maintenance Range | 1mg-2.5mg per week | maintenance | Typical maintenance dose range |
| Week 13+ | 1.0–2.0 mg | maintenance | Individualize. Max clinical dose 2.4 mg/week. |
- Semaglutide se suministra como polvo liofilizado.
- Semaglutide debe reconstituirse con agua bacteriostática antes de su uso.
- Elija el volumen de reconstitución según el tamaño del vial para facilitar la dosificación.
| Dose | Units to Draw | Volume (mL) | Approx. Supply |
|---|---|---|---|
| 0.25mg | 5 units | - | 20 weeks |
| 0.5mg | 10 units | - | 10 weeks |
| 0.75mg | 15 units | - | 6-7 weeks |
| 1mg | 20 units | - | 5 weeks |
| 1.25mg | 25 units | - | 4 weeks |
| 1.5mg | 30 units | - | 3 weeks |
| 1.75mg | 35 units | - | 3 weeks |
| 2mg | 40 units | - | 2.5 weeks |
| 2.5mg | 50 units | - | 2 weeks |
Identity
- Name: Semaglutide
- Product Type: Vial | Subcutaneous Injection
- CAS Number: 910463-68-2
- Available Strengths: 5mg, 10mg, 15mg, 20mg, 30mg
- Molecular Formula: C₁₈₇H₂₉₁N₄₅O₅₉
- Molecular Weight: 4,113.6 Da
- Sequence / Type: GLP-1 Receptor Agonist
- Available Strengths: 5mg, 10mg, 15mg, 20mg, 30mg, 100mg
Quality & Purity
- Purity: 99%+
- Purity: ≥ 99%
- Endotoxin: ≤ 1 EU/mg
- Appearance: White lyophilized powder
- Solubility: Bacteriostatic water
Storage & Handling
- Storage: Refrigerate after reconstitution (2-8°C)
- Pre-use Storage: -20°C (long-term) / 2–8°C (short)
- Post-Reconstitution: 2–8°C · Up to 28 days
- Shelf Life: 18 months from manufacture
Timing: Use consistent administration timing for stable protocol tracking.
Storage: Refrigerate 2–8°C · 18-month shelf life
Frequency: StartingDose:O.25mg onceweekly
Cycle: Titration:Increasegraduallyby0.25-0.5mgevery2-4weeks
Injection Sites: Rotate approved injection sites to reduce local irritation risk.