Visceral fat reduction, muscle tone improvement, anti-aging, lean body mass development, fat loss, metabolic marker improvement
Tesamorelin es un péptido sintético que estimula la liberación de la hormona del crecimiento (GH) actuando como un análogo de la hormona liberadora de la hormona del crecimiento (GHRH). Originalmente aprobado por FDA para la lipodistrofia relacionada con el VIH, ahora se usa ampliamente de forma no autorizada para reducir la grasa visceral, mejorar el tono muscular y apoyar el antienvejecimiento. Tesamorelin promueve el desarrollo de masa corporal magra, la pérdida de grasa y la mejora de los marcadores metabólicos.
Mechanism of Action - Growth Hormone Peptides Pathway
Dosis típica:0,5-1 mg por día (hasta 3 veces por día)
Frecuencia:Diaria, matutina o nocturna.(Se puede tomar mañana, tarde y noche)
Ciclo:De forma continua o en bloques de 8 a 12 semanas
| Period | Dose | Phase | Clinical Notes |
|---|---|---|---|
| Typical Dose | 0.5-1mg per day (up to 3x per day) | maintenance | Daily, Morning or Nighttime. Ongoing or in 8-12 week blocks. |
| Week 5+ | 2 mg | maintenance | Full clinical dose. Monitor GH and IGF-1 levels. |
- Tesamorelin se suministra como polvo liofilizado.
- Tesamorelin debe reconstituirse con agua bacteriostática antes de su uso.
- El volumen de reconstitución varía ligeramente según el tamaño del vial para mantener una dosificación sencilla.
| Dose | Units to Draw | Volume (mL) | Approx. Supply |
|---|---|---|---|
| 0.5mg | 10 units | - | 10 doses (1+ week) |
| 1mg | 20 units | - | 5 doses (0.5 week) |
| 2mg | 40 units | - | 2-3 doses |
| Dose | Units to Draw | Volume (mL) | Approx. Supply |
|---|---|---|---|
| 0.5mg | 10 units | - | 20 doses (2+ weeks) |
| 1mg | 20 units | - | 10 doses (1+ weeks) |
| 2mg | 40 units | - | 5 doses (0.5 weeks) |
| Dose | Units to Draw | Volume (mL) | Approx. Supply |
|---|---|---|---|
| 0.5mg | 10 units | - | 30 doses (3+ weeks) |
| 1mg | 20 units | - | 15 doses (2+ weeks) |
| 2mg | 40 units | - | 7 doses (1 week) |
| Dose | Units to Draw | Volume (mL) | Approx. Supply |
|---|---|---|---|
| 0.5mg | ~7.5 units | - | 40 doses (4+ weeks) |
| 1mg | ~15 units | - | 20 doses (3 weeks) |
| 2mg | ~30 units | - | 10 doses (1.5 weeks) |
Identity
- Name: Tesamorelin
- Product Type: Vial | Subcutaneous Injection
- CAS Number: 218949-48-5
- Available Strengths: 5mg, 10mg, 15mg, 20mg
- Molecular Formula: C₂₂₁H₃₆₆N₇₂O₆₄S
- Molecular Weight: 5,135.8 Da
- Sequence / Type: GHRH analogue (1–44)
- Available Strengths: 5mg, 10mg
Quality & Purity
- Purity: 99%+
- Purity: ≥ 99%
- Endotoxin: ≤ 1 EU/mg
- Appearance: White lyophilized powder
- Solubility: Bacteriostatic water
Storage & Handling
- Storage: Refrigerate after reconstitution (2-8°C)
- Pre-use Storage: -20°C (long-term) / 2–8°C (short)
- Post-Reconstitution: 2–8°C · Up to 28 days
- Shelf Life: 18 months from manufacture
Timing: Daily,Morning or Nightime. (Canbetakenmorning,afternoon,nighttime)
Storage: Refrigerate 2–8°C · 18-month shelf life
Frequency: Frequency: Daily,Morning or Nightime.
Cycle: Ongoing or in 8-12 week blocks
Injection Sites: Rotate approved injection sites to reduce local irritation risk.